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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T10665 | Calcium-Sensing Receptor Antagonists I | Others | |
Calcium-Sensing Receptor Antagonists I functions as an antagonist to the parathyroid hormone receptors that sense calcium. | |||
T22795 | Gadolinium chloride | CaSR | |
Gadolinium chloride is a calcium-sensing receptor (CaSR) agonist | |||
T3802 | Ligustroflavone | Nuezhenoside | Others , CaSR |
Ligustroflavone (Nuezhenoside) has anti-inflammatory activity. | |||
T12846 | SB-423562 | CaSR | |
SB-423562 is a calcium-sensing receptor (CaSR) antagonist and can be used in studies about osteoporosis. | |||
T8457 | NPS2390 | GluR | |
NPS2390 is a first generation quinoxaline derivative that acts as a noncompetitive antagonist of mGluR1 and mGluR5 (IC50 of 5.2 and 82 nM, respectively) | |||
T15261 | Evocalcet | KHK7580 | CaSR |
Evocalcet (KHK7580) has an activating effect on the calcium-sensing receptor (CaSR). | |||
T8403 | Cinacalcet | AMG 073 | CaSR |
Cinacalcet (AMG 073) is an orally active, allosteric Ca receptor (CaR) agonist, treatment of cardiovascular disease . | |||
T1641 | Strontium ranelate | Distrontium renelate,S12911 | Calcium Channel , CaSR |
Strontium ranelate (S12911), a strontium (II) salt of the ranelic acid, is a medication for osteoporosis. Studies indicate it can also slow the course of osteoarthritis of the knee. The drug is unusual in that it both in... | |||
T2406 | Cinacalcet hydrochloride | AMG-073 HCl,Cinacalcet HCl,AMG-073 hydrochloride,Cinacalcet | CaSR |
Cinacalcet hydrochloride (AMG-073 hydrochloride) is a naphthalene derivative and CALCIMIMETIC AGENT that increases the sensitivity of PARATHYROID GLAND calcium-sensing receptors to serum calcium. This action reduces para... | |||
TP1236 | Etelcalcetide hydrochloride | AMG 416 hydrochloride,KAI-4169 hydrochloride | CaSR |
Etelcalcetide hydrochloride (AMG 416 hydrochloride) is a synthetic peptide that acts as an allosteric modulator of the calcium-sensing receptor (CaSR), effectively lowering parathyroid hormone (PTH) levels in patients wi... | |||
T1730 | NPS-2143 | SB262470,NPS 2143,SB 262470A | Calcium Channel , CaSR |
NPS-2143 (SB 262470A) is a novel potent and selective antagonist of Ca(2+) receptor. | |||
T4967 | NPS-2143 hydrochloride | NPS-2143 HCL | CaSR |
NPS-2143 hydrochloride (NPS-2143 HCL) is a selective potent calcium ion-sensing receptor antagonist. | |||
T23401 | Strontium chloride | Others , CaSR | |
Strontium chloride is an agonist of Calcium sensing receptor (CaSR) and directly affects C-type nerve fibers. | |||
T13918 | Tecalcet Hydrochloride | R-568 hydrochloride,R-568 (hydrochloride) | CaSR |
Tecalcet Hydrochloride (R-568 hydrochloride) is an allosteric and positive modulator of the calcium-sensing receptor(CaSR). Tecalcet Hydrochloride increases the sensitivity to the activation of extracellular Ca2+. | |||
T28691 | SB-423562 HCl | SB-423562,SB-423562A,SB-423562-A,NPSP795,NPSP-795,SHP-635 | |
SB-423562 is a calcium-sensing receptor antagonist. | |||
T28870 | Strontium Malonate | NBS-101,NBS 101,NBS101 | |
Strontium Malonate, a calcium-sensing receptor agonist, is used potentially for the treatment of postmenopausal osteoporosis. | |||
T31624 | Encaleret | JIT305,JIT 305 | |
Encaleret( JIT-305) is an antagonist of oral calcium-sensing receptor (CaSR), it is used for the treatment of osteoporosis. | |||
T72908 | Gamma-Glu-Abu | ||
Gamma-Glu-Abu is a potent calcium sensing receptor (CaSR) agonist . | |||
T12845 | SB-423557 | Calcium Channel | |
SB-423557 is an orally active antagonist of calcium-sensing receptor (CaR) with IC50 of 520 nM | |||
T21758 | Calindol (hydrochloride) | ||
Calindol (hydrochloride) is a positive allosteric modulator (PAM) of calcimimetic calcium-sensing receptor (CaSR) with an EC50 of 132 nM. |